In vivo pharmacokinetics
-In vivo absorption assay
-Tissue distribution
-Material balance
In vitro pharmacokinetics
-Cell permeability test (caco-2 cells, MDCK cells)
-Plasma protein binding test
-Whole blood plasma partition ratio test
-Metabolic stability studies in hepatocytes/hepatic microsomes/lung microsomes/lung S9
-Metabolite identification studies in hepatocytes/hepatic microsomes/lung microsomes/lung S9
-In vivo metabolite identification (blood, urine, feces, bile, lung tissue, etc.)
-CYP reversible inhibition/time-dependent inhibition assay
-CYP metabolic phenotyping assays
-CYP enzyme induction assay
-ABC transporter assay (caco-2 cells)
-SLC transporter assay (HEK293 cells)
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